5lma A 1.43 BS01 6ZG A 1 L377 A400 M450 A451 G454 P455 R498 L501 D512 L15 A38 M88 A89 G92 P93 R136 L139 D150 D494 A496 R498 N499 D512 K533 D132 A134 R136 N137 D150 K169 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.25uM -logKd/Ki=6.60, IC50=0.25uM IC50=2512nM P43405 27578246 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYD