5kbr A 2.36 BS01 IPW A 1 I276 V284 A297 K299 V328 V342 M344 E345 Y346 L347 L396 T406 I22 V30 A36 K38 V58 V66 M68 E69 Y70 L71 L120 T130 N389 K391 D393 N394 D407 T427 N113 K115 D117 N118 D131 T144 2.7.11.1 0004672,0005524,0006468 ic50=260nM -logKd/Ki=6.59, IC50=260nM Q13153 27994749 601 EKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAEVAIKQELIINEILVMRENKNPNIVNYLDSYWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLDMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK