5kbq A 2.58 BS01 IPV A 1 I276 G277 Q278 V284 A297 K299 E315 V342 M344 Y346 L347 L396 T406 I23 G24 Q25 V31 A44 K46 E62 V89 M91 Y93 L94 L143 T153 N389 K391 D393 N394 D407 P416 T427 N136 K138 D140 N141 D154 P163 T174 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.00, IC50=100nM IC50=100nM Q13153 27994749 601 LEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSEMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLDMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATK