5k13 A 1.85 BS01 6Q7 A 1 W225 F228 S232 C235 L266 L269 I270 I273 F286 S287 G301 F302 V395 P407 W45 F48 S52 C55 L86 L89 I90 I93 F106 S107 G121 F122 V215 P227 ? 0003677,0004879,0005634,0006355,0048384 Ki=1.8nM -logKd/Ki=8.74, Ki=1.8nM Ki=1.8nM P10276 27261179 501 TPEVGELIEKVRKAHQETFPALCQLGKYTTNNSSEQRVSLDIDLWDKFSELSTKCIIKTVEFAKQLPGFTTLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFAFANQLLPLEMDDAETGLLSAICLICGDRQDLEQPDRVDMLQEPLLEALKVYVRKRRPSRPHMFPKMLMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLE