5k00 A 1.77 BS01 6PV A 1 A38 K40 L61 L64 C70 L86 Y88 C89 G92 E93 L139 I149 D150 F151 A35 K37 L58 L61 C67 L83 Y85 C86 G89 E90 L136 I146 D147 F148 D132 K134 E136 N137 D150 S171 D129 K131 E133 N134 D147 S155 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=7nM -logKd/Ki=8.15, IC50=7nM Q14680 28186750 401 MDYDELLKYYELHETIGTGAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARG