5jsm A 2.19 BS01 6NB B 1 Q461 I463 V471 A481 K483 L514 F516 T529 Q530 W531 C532 S535 H539 F583 D594 F595 G596 Q17 I19 V27 A37 K39 L70 F72 T85 Q86 W87 C88 S91 H95 F139 D150 F151 G152 D576 K578 N580 N581 D594 S616 D132 K134 N136 N137 D150 S160 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=6.59, IC50=260nM P15056 27571413 801 SEFDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHASETKFEMKKLIDIARQTARGMDYLHAKSIIHRDLKSNNIFLHEDNTVKIGDFGLATEKSGSILWMAPEVIRMQDSNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIEMVGRGSLSPDLSKVRSNCPKRMKRLMAECLKKKRDERPSFPRILAEIEELAREL