5jkg A 2.352 BS01 6LF A 1 L473 E475 E551 C552 A553 G556 N557 R616 L619 L21 E23 E96 C97 A98 G101 N102 R149 L152 D612 A614 R616 N617 D630 D145 A147 R149 N150 D163 2.7.10.1 0004672,0004713,0005524,0006468 ic50<6.4nM IC50=6.0nM P22455 27618313 801 DLPLDPLWEFPRDRLVLGKPLGEGAFGQVVRAEAFGMDPARPDQASTVAVKMLKDDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPGPPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV