5i9i A 2.7 BS01 5HV A 1 F110 L111 L121 G152 L153 G154 L159 S273 F274 W298 H351 Q352 F357 L369 L371 F57 L58 L68 G99 L100 G101 L106 S220 F221 W245 H298 Q299 F304 L316 L318 3.1.1.47 0003847,0005515,0005543,0005576,0009395,0016486,0016787,0016788,0034362,0034364,0034374,0034440,0034441,0034638,0046469,0047499,0050729,0062234,0090026 -logKd/Ki=7.30, Kd=49.7nM IC50=0.250000nM, Ki=110nM, Kd=5.0nM Q13093 27078579 501 TKIPRGNGPYSVGCTDLMFDHTNKGTFLRLYYPSQDNDRLDTLWIPNKEYFWGLSKFLGTHWLMGNILRLLFGSMTTPANWNSPLRPGEKYPLVVFSHGLGAFRTLYSAIGIDLASHGFIVAAVEHRDRSASATYYFKDQSAAEIGDKSWLYLRTLKQEEETHIRNEQVRQRAKECSQALSLILDIDHGKPVKNALDLKFDMEQLKDSIDREKIAVIGHSFGGATVIQTLSEDQRFRCGIALDAWMFPLGDEVYSRIPQPLFFINSEYFQYPANIIKMKKCYSPDKERKMITIRGSVHQNFADFTFATGKIIGHMLKLKGDIDSNVAIDLSNKASLAFLQKHLGLHKDFDQWDCLIEGDDENLIPGTNINT