5i12 A 1.59 BS01 ZN A 1 H226 H230 H236 H114 H118 H124 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 27356908 301 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5i12 A 1.59 BS02 ZN A 2 H175 D177 H190 H203 H63 D65 H78 H91 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 27356908 302 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5i12 A 1.59 BS03 CA A 1 D182 G183 D185 L187 D205 E208 D70 G71 D73 L75 D93 E96 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 27356908 303 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5i12 A 1.59 BS04 CA A 2 D165 G197 Q199 D201 D53 G85 Q87 D89 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 27356908 304 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5i12 A 1.59 BS05 CA A 3 D131 D206 E208 D19 D94 E96 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 27356908 305 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 5i12 A 1.59 BS06 H27 A 1 L187 A189 H226 E227 H230 H236 Y245 P246 M247 Y248 L75 A77 H114 E115 H118 H124 Y133 P134 M135 Y136 H226 E227 H230 H236 H114 E115 H118 H124 3.4.24.35 0004222,0006508,0008237,0008270,0031012 ic50=1200nM -logKd/Ki=5.92, IC50=1200nM P14780 27356908 306 DLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGVGYSLFLVAAHEFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG