5h0h A 1.72 BS01 OOV A 1 L273 A275 V281 A293 K295 V323 L325 T338 M341 D348 L393 D404 F405 L189 A191 V197 A209 K211 V239 L241 T254 M257 D264 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=686nM -logKd/Ki=6.16, IC50=686nM IC50=692nM P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP