5h0g A 1.8 BS01 OOU A 1 L273 V281 A293 K295 V323 T338 M341 S345 D348 A390 L393 D404 F405 L189 V197 A209 K211 V239 T254 M257 S261 D264 A306 L309 D320 F321 D386 R388 A390 N391 D404 F424 D302 R304 A306 N307 D320 F340 2.7.10.2 0004672,0004713,0005524,0006468 ic50=111nM -logKd/Ki=6.95, IC50=111nM IC50=111nM P08631 28662963 601 RIIVVALYDYEAIHHEDLSFQKGDQMVVLEESGEWWKARSLATRKEGYIPSNYVARVDSLETEEWFFKGISRKDAERQLLAPGNMLGSFMIRDSETTKGSYSLSVRDYDPRQGDTVKHYKIRTLDNGGFYISPRSTFSTLQELVDHYKKGNDGLCQKLSVPCMSSKPQKPWEKDAWEIPRESLKLEKKLGAGQFGEVWMATYNKHTKVAVKTMKPGSMSVEAFLAEANVMKTLQHDKLVKLHAVVTKEPIYIITEFMAKGSLLDFLKSDEGSKQPLPKLIDFSAQIAEGMAFIEQRNYIHRDLRAANILVSASLVCKIADFGLARVIEDNEYTAREGAKFPIKWTAPEAINFGSFTIKSDVWSFGILLMEIVTYGRIPYPGMSNPEVIRALERGYRMPRPENCPEELYNIMMRCWKNRPEERPTFEYIQSVLDDFYTATESQYEEIP