5gjf A 2.89 BS01 6V4 A 1 V42 V50 A61 E77 L81 V90 M104 Y106 A107 L163 C174 D175 V17 V25 A36 E47 L51 V60 M74 Y76 A77 L133 C144 D145 D156 K158 P160 N161 I173 D175 M186 D126 K128 P130 N131 I143 D145 M156 2.7.11.25 0000287,0004672,0004709,0005524,0006468,0007165 -logKd/Ki=6.59, IC50=260nM O43318,Q15750 27803473 601 GPLHMIDYKEIEVEEVVGRGAFGVVCKAKWRAKDVAIKQIRKAFIVELRQLSRVNHPNIVKLYGACLNPVCLVMEYAEGGSLYNVLHGAEPLPYYTAAHAMSWCLQCSQGVAYLHSMQPKALIHRDLKPPNLLLVAGGTVLKICDFGTACDIQTHMTNNKGSAAWMAPEVFEGSNYSEKCDVFSWGIILWEVITRRKPFDEIGGPAFRIMWAVHNGTRPPLIKNLPKPIESLMTRCWSKDPSQRPSMEEIVKIMTHLMRYFPGADEPLQYPCQHSLPGRVEPYVDFAEFYRLWSVDHG