5fxr A 2.4 BS01 8LN A 1 L1005 V1013 A1031 M1079 M1082 G1085 M1156 L26 V34 A52 M99 M102 G105 M176 D1135 R1139 N1140 D1153 E1162 D155 R159 N160 D173 E182 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 -logKd/Ki=7.42, IC50=0.038uM IC50=38nM P08069 27078757 2284 GYFSADVYVPDEWEVAREKITMSRELGQGSFGMVYEGVAKGVVKDEPETRVAIKTVEAASMRERIEFLNEASVMKEFNCHHVVRLLGVVSQGQPTLVIMELMTRGDLKSYLRSLRPEMENNPVLAPPSLSKMIQMAGEIADGMAYLNANKFVHRDLAARNCMVAEDFTVKIGDFGMTRDIYETDYYRKGLLPVRWMSPESLKDGVFTTYSDVWSFGVVLWEIATLAEQPYQGLSNEQVLRFVMEGGLLDKPDNCPDMLFELMRMCWQYNPKMRPSFLEIISSIKEEMEPGFREVSFYYSE