5dls A 2.15 BS01 5CV A 1 G18 G21 A36 K38 E85 Y86 C87 G90 L137 D148 G13 G16 A31 K33 E72 Y73 C74 G77 L124 D135 D130 K132 E134 N135 D148 T170 D117 K119 E121 N122 D135 T157 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=4.4nM -logKd/Ki=8.36, IC50=4.4nM O14757 26437226 301 VEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK