5cy3 A 1.76 BS01 55Y A 1 L377 V385 A400 K402 M448 A451 G454 L501 S511 D512 L18 V26 A41 K43 M87 A90 G93 L140 S150 D151 D494 A496 R498 N499 D512 K533 D133 A135 R137 N138 D151 K172 2.7.10.2 0004672,0004713,0005524,0006468 ic50=16nM -logKd/Ki=7.80, IC50=16nM IC50=16nM P43405 26320624 701 PKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVTDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEG