5bqi A 1.88 BS01 4UL A 1 A123 P124 S127 V128 A119 P120 S123 V124 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 ic50=0.9nM -logKd/Ki=9.05, IC50=0.9nM O14684 26653180 201 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL 5bqi A 1.88 BS02 GSH A 1 N74 E77 H113 Y117 R126 S127 Y130 N70 E73 H109 Y113 R122 S123 Y126 1.11.1.-,2.5.1.18,5.3.99.3 0001516,0004364,0004602,0004667,0005515,0005641,0005737,0005789,0006693,0007165,0008283,0008285,0016020,0016491,0016740,0016853,0019233,0031620,0032308,0043295,0048471,0050220,0050727,0098869 O14684 26653180 202 SLVMSSPALPAFLLCSTLLVIKMYVVAIITGQVRLRKKAFANPEDALRHGGPQYCRSDPDVERCLRAHRNDMETIYPFLFLGFVYSFLGPNPFVAWMHFLVFLVGRVAHTVAYLGKLRAPIRSVTYTLAQLPCASMALQILWEAARHL