5av0 A 1.85 BS01 47X A 1 V27 A40 E94 L95 E100 I160 V26 A39 E93 L94 E99 I158 D139 K141 E143 N144 D161 T180 D137 K139 E141 N142 D159 T178 2.7.11.1 0004672,0005524,0006468 ic50=280uM -logKd/Ki=3.55, IC50=280uM IC50=280000nM P53355 26322379 300 TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKSLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKP