4zy4 A 2.6 BS01 4T3 A 1 A297 E345 Y346 L347 A348 G350 L396 A49 E92 Y93 L94 A95 G97 L143 N389 K391 D393 N394 D407 P416 T427 N136 K138 D140 N141 D154 P163 T174 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.66, Ki=22nM Ki=22nM Q13153 26030457 601 SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIKQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRNIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT