4yp8 A 2.641 BS01 4GF A 1 M192 G193 E194 V200 A211 Y262 Y264 M265 P266 G268 S269 L318 M29 G30 E31 V37 A48 Y94 Y96 M97 P98 G100 S101 L150 D311 K313 A315 N316 D329 T351 D143 K145 A147 N148 D161 T179 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 -logKd/Ki=7.89, IC50=13nM IC50=13nM Q9NWZ3 26101573 501 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLATTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASETVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA