4xg3 A 2.3 BS01 X3G A 1 L377 V385 A400 M448 M450 A451 G454 P455 K458 R498 L501 D512 L15 V18 A33 M76 M78 A79 G82 P83 K86 R126 L129 D140 D494 A496 R498 N499 D512 K533 D122 A124 R126 N127 D140 K161 2.7.10.2 0004672,0004713,0005524,0006468 ic50=17.5nM -logKd/Ki=7.76, IC50=17.5nM P43405 27504936 701 VYLDRKLLTLEDKELGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVV