4rj7 A 2.55 BS01 3R1 A 1 L718 F723 V726 A743 K745 M793 G796 L844 L22 F27 V30 A47 K49 M92 G95 L143 D837 A839 R841 N842 D855 D136 A138 R140 N141 D154 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=7.66, Ki=22nM Ki=101nM P00533 25383627 1102 EAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKESPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGRAKLVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFDMDDVVDADEYLI