4rak A 2.04 BS01 652 A 1 F271 T272 L274 A275 S278 M312 T316 R319 F329 L330 L345 I353 F54 T55 L57 A58 S61 M95 T99 R102 F112 L113 L128 I136 ? 0003677,0004879,0006629 Ki=14nM -logKd/Ki=7.85, Ki=14nM EC50=250nM, Ki=14nM P55055 25435151 503 VQLTAAQELMIQQLVAAQLQCNKRSFSDQPKVTPWPLGADPQSRDARQQRFAHFTELAIISVQEIVDFAKQVPGFLQLGREDQIALLKASTIEIMLLETARRYNHETECITFLKDFTYSKDDFHRAGLQVEFINPIFEFSRAMRRLGLDDAEYALLIAINIFSADRPNVQEPGRVEALQQPYVEALLSYTRIKRPQDQLRFPRMLMKLVSLRTLSSVHSEQVFALRKLPPLLSEIW