4ra5 A 2.61 BS01 3L0 A 1 L386 G387 K388 V394 A407 M458 E459 D508 L511 D522 F664 F668 L13 G14 K15 V21 A34 M85 E86 D135 L138 D149 F291 F295 D504 K506 D508 N509 D522 T542 D131 K133 D135 N136 D149 T169 2.7.11.13 0004672,0004674,0004697,0005524,0006468 -logKd/Ki=8.40, IC50=4nM IC50=4.0nM Q04759 25254961 801 KLKIEDFELHKMLGKGSFGKVFLAEFKKTNQFFAIKALKKDVVLMDDDVECTMVEKRVLSLAWEHPFLTHMFCTFQTKENLFFVMEYLNGGDLMYHIQSCHKFDLSRATFYAAEIILGLQFLHSKGIVYRDLKLDNILLDKDGHIKIADFGMCKENMLGDAKTNEFCGTPDYIAPEILLGQKYNHSVDWWSFGVLLYEMLIGQSPFHGQDEEELFHSIRMDNPFYPRWLEKEAKDLLVKLFVREPEKRLGVRGDIRQHPLFREINWEELERKEIDPPFRPKVKSPFDCSNFDKEFLNEKPRLSFADRALINSMDQNMFRNFSFMNPGMERLISH