4r2u A 2.3 BS01 3JX A 1 F282 G284 C285 Q286 R288 S289 H323 I326 Y327 L330 I341 S342 M364 H449 Y473 F66 G68 C69 Q70 R72 S73 H107 I110 Y111 L114 I125 S126 M148 H233 Y257 ? 0003677,0004879,0005634,0006355 IC50=80nM, EC50=4288nM P37231 26068133 501 NPESADLRALAKHLYDSYIKSFPLTKAKARAILTGTDKSPFVIYDMNSLMMGEDKIKSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL