4qyg A 1.75 BS01 3DW A 1 L15 A36 K38 L84 Y86 C87 L137 D148 L13 A34 K36 L75 Y77 C78 L128 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.0041uM -logKd/Ki=8.39, IC50=4.1nM IC50=>10000nM O14757 25453805 301 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA