4qt1 A 2.4 BS01 3C9 A 1 L828 G829 K830 V836 A853 Y904 L905 L956 L15 G16 K17 V23 A40 Y85 L86 L137 D949 A951 R953 N954 D967 D130 A132 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 ic50=7nM -logKd/Ki=8.15, IC50=7nM IC50=7.0nM P52333 25262541 1201 PTIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDMLWSGS