4qq5 A 2.203 BS01 37O A 1 L478 E480 C482 F483 E525 I539 L555 C557 A558 A559 G561 L624 D635 F636 L32 E34 C36 F37 E74 I88 L104 C106 A107 A108 G110 L160 D171 F172 D617 A619 R621 N622 D635 D153 A155 R157 N158 D171 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.32, IC50=482nM P22455 25317566 801 QDPLLAGLVSLDLPLDPLWEFPRDRLVLGKPLGEGCFGQVVRAEAFGMDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVILECAAKGNLREFLRARRPPGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLALPVKWMAPEALFDEVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV