4puj A 1.42 BS01 ZN A 1 C318 C320 C323 H349 C302 C304 C307 H333 D102 D280 C318 C320 C323 H349 D93 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0016763,0046872,0101030 P28720 24955548 401 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA 4puj A 1.42 BS02 CKR A 1 D102 Y106 D156 C158 G229 L231 A232 M260 G261 R286 D93 Y97 D140 C142 G213 L215 A216 M244 G245 R270 D102 D280 C318 C320 C323 H349 D93 D264 C302 C304 C307 H333 2.4.2.29 0002099,0005737,0005829,0006400,0008033,0008479,0008616,0016757,0016763,0046872,0101030 Kd=35nM -logKd/Ki=7.46, Kd=35.0nM P28720 24955548 407 DRPRFSFSIAAREGKARTGTIEMKRGVIRTPAFMPVGTAATVKALKPETVRATGADIILGNTYHLMLRPGAERIAKLGGLHSFMGWDRPILTDSGGYQVMSLLTKQSEEGVTFKSRHMLSPERSIEIQHLLGSDIVMAFDECTPYPATPSRAASSMERSMRWAKRSRDAFDSRKEQAENAALFGIQQGSVFENLRQQSADALAEIGFDGYAVGGLAVGEGQDEMFRVLDFSVPMLPDDKPHYLMGVGKPDDIVGAVERGIDMFDCVLPTRSGRNGQAFTWDGPINIRNARFSEDLKPLDSECHCAVCQKWSRAYIHHLIRAGEILGAMLMTEHNIAFYQQLMQKIRDSISEGRFSQFAQDFRARYFA