4oth A 1.8 BS01 DRN A 1 G628 F632 A648 K650 M701 S704 D708 D750 L753 A763 D764 F910 G17 F21 A37 K39 M90 S93 D97 D139 L142 A152 D153 F270 D746 K748 D750 N751 D764 D135 K137 D139 N140 D153 2.7.11.13 0004672,0004674,0005524,0006468 ic50=9nM -logKd/Ki=8.05, IC50=9nM Q16512 25111382 1001 RKSPLTLEDFKFLAVLGRGHFGKVLLSEFRPSGELFAIKALKKGDIVARDEVESLMCEKRILAAVTSAGHPFLVNLFGCFQTPEHVCFVMEYSAGGDLMLHIHSDVFSEPRAIFYSACVVLGLQFLHEHKIVYRDLKLDNLLLDTEGYVKIADFGLCKTRAVDWWGLGVLLYEMLVGESPFPGDDEEEVFDSIVNDEVRYPRFLSAEAIGIMRRLLRRNPERRLGSSERDAEDVKKQPFFRTLGWEALLARRLPPPFVPTLSGRTDVSNFDEEFTGEAPTLSPPRDARPLTAAEQAAFLDFDFVAG