4n7u A 1.4598 BS01 2JA A 1 R412 R418 R469 R116 R122 R173 ? Kd=0.51uM -logKd/Ki=6.29, Kd=0.51uM IC50=7870nM, EC50=2.0nM O00481 24703779 501 GAYNEWKKALFKPADVILDPKTADPILLVSEDQRSVERAKEPQDLPDNPERFNWHYCVLGCESFISGRHYWEVEVGDRKEWHIGVCSKNVQRKGWVKMTPENGFWTMGLTDGNKYRTLTEPRTNLKLPKPPKKVGVFLDYETGDISFYNAVDGSHIHTFLDVSFSEALYPVFRILTLEPTALTICP