4lgh A 2.84 BS01 0JN A 1 L273 A293 K295 M314 I336 G338 Y340 M341 L393 L17 A34 K36 M43 I65 G67 Y69 M70 L122 D386 R388 A390 N391 D404 D115 R117 A119 N120 D133 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.70, IC50=2nM IC50=620nM P00523 23841803 601 KDAWEIPRESLRLEVKLGQGGEVWMGTWNGTRVAIKTLEAQVMKKLRHEKLVQLYAVVSEEPIYIVGEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL