4l9i A 2.32 BS01 8PR A 1 R195 V201 A214 T265 M267 D271 E318 L321 R166 V172 A185 T236 M238 D242 E289 L292 D314 K316 E318 N319 D332 A341 T352 D285 K287 E289 N290 D303 A312 T323 2.7.11.14 0001750,0004672,0004674,0004703,0005515,0005524,0005737,0006468,0007165,0007601,0009966,0016020,0016310,0022400,0042995,0046777,0050254,0097381 Kd=13uM -logKd/Ki=4.89, Kd=13uM IC50=398100nM P28327 24220010 601 SRDRKYLARLKLPPLSKCEALRESLDLGFEGMCLEQPIGKRLFQQFLRTHEQHGPALQLWKDIEDYDTADDALRPQKAQALRAAYLEPQAQLFCSFLDAETVARARAGAGDGLFQPLLRAVLAHLGQAPFQEFLDSLYFLRFLQWKWLEAQPMGEDWFLDFRVLGRGGFGEVFACQMKATGKLYACKKLNKKRLKKRKGYQGAMVEKKILAKVHSRFIVSLAYAFETKTDLCLVMTIMNGGDIRYHIYNVDEDNPGFQEPRAIFYTAQIVSGLEHLHQRNIIYRDLKPENVLLDDDGNVRISDLGLAVELKAGQTKTKGYAGTPGFMAPELLLGEEYDFSVDYFALGVTLYEMIAARGPFRARGEKVENKELKQRVLEQAVTYPDKFSPASKDFCEALLQKDPEKRLGFRDGSCDGLRTHPLFRDISWRQLEAGMLTPPFVPDSRTVYAKNIQDVGAFSTVKGVAFEKADTEFFQEFASGTCPIPWQEEMIETGVFGDLNVWRP