4l43 A 3.0 BS01 5FI A 1 G75 G77 Y79 G80 V82 A98 L102 E150 Y151 L152 M202 D213 K218 G18 G20 Y22 G23 V25 A41 L45 E93 Y94 L95 M145 D156 K161 D195 K197 E199 N200 D213 T233 D138 K140 E142 N143 D156 T165 2.7.11.1 0004672,0004674,0005524,0006468 Ki=20nM, IC50=160nM P23443 23731517 401 RGPEKIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLLQSEEDVSQFDSKFTRQTPVSANQVFLGFAYVAPS