4kqs A 1.97 BS01 MG A 1 D103 D107 D90 D94 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F85 D90 D94 R99 D161 K187 F226 D230 D231 2.5.1.1,2.5.1.10 0004659,0008299,0016765 P14324 401 VYAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFASFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4kqs A 1.97 BS02 MG A 2 D103 D107 D90 D94 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F85 D90 D94 R99 D161 K187 F226 D230 D231 2.5.1.1,2.5.1.10 0004659,0008299,0016765 P14324 402 VYAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFASFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4kqs A 1.97 BS03 IPE A 1 K57 R60 Q96 R113 F239 K44 R47 Q83 R100 F226 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F85 D90 D94 R99 D161 K187 F226 D230 D231 2.5.1.1,2.5.1.10 0004659,0008299,0016765 P14324 404 VYAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFASFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK 4kqs A 1.97 BS04 RIS A 1 D103 R112 Q171 K200 T201 D243 K257 D90 R99 Q158 K187 T188 D230 K244 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K44 F85 D90 D94 R99 D161 K187 F226 D230 D231 2.5.1.1,2.5.1.10 0004659,0008299,0016765 IC50=11nM, Ki=82.2nM P14324 405 VYAQEKQDFVQHFSQIVRVLTEPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFASFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYKRRK