4kio A 2.18 BS01 G5K A 1 I369 A389 F435 F437 M438 G441 C442 L489 I15 A32 F72 F74 M75 G78 C79 L126 D482 A484 R486 N487 D500 P521 D119 A121 R123 N124 D137 P142 2.7.10.2 0004672,0004713,0004715,0005524,0006468 ic50=0.5uM -logKd/Ki=6.30, IC50=0.501uM Q08881 23935099 701 GSVIDPSELTFVQEIGSGLVHLGYWLNKDKVAIKTIEEDFIEEAEVMMKLSHPKLVQLYGVCLEQAPICLVFEFMEHGCLSDYLRTQRGLFAAETLLGMCLDVCEGMAYLEEACVIHRDLAARNCLVGENQVIKVSDFGMTPVKWASPEVFSFSRYSSKSDVWSFGVLMWEVFSEGKIPYENRSNSEVVEDISTGFRLYKPRLASTHVYQIMNHCWKERPEDRPAFSRLLRQLAEIAESG