4kbk A 2.1 BS01 1QG A 1 I15 I23 A36 K38 M80 M82 L85 G86 L135 I148 I13 I19 A32 K34 M70 M72 L75 G76 L125 I138 D128 K130 D118 K120 2.7.11.1,2.7.11.26 0004672,0005524,0006468 -logKd/Ki=8.18, IC50=6.6nM IC50=6.6nM P48730 23919824 401 LRVGNRYRLGRKIGSGGDIYLGTDIAAGEEVAIKLECQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML