4kb8 A 1.95 BS01 1QN A 1 I23 A36 K38 M80 M82 L85 G86 L135 I148 I21 A34 K36 M78 M80 L83 G84 L133 I146 D128 K130 D126 K128 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=12.9nM -logKd/Ki=7.89, IC50=12.9nM IC50=64nM P48730 23919824 401 LRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNML