4iw0 A 4.0 BS01 BX7 A 1 L15 G16 Q17 G18 A21 V23 A36 F88 C89 G92 M142 D157 L16 G17 Q18 G19 A22 V24 A37 F89 C90 G93 M143 D158 N135 K137 N140 D157 T176 N136 K138 N141 D158 T177 2.7.11.1 0002218,0002753,0003676,0004672,0004674,0005515,0005524,0005654,0005737,0005829,0006338,0006468,0006954,0007249,0009615,0010468,0010508,0010628,0010629,0016236,0016239,0016310,0018105,0018107,0019903,0032479,0032481,0032727,0032728,0033138,0034142,0042802,0043123,0043231,0044024,0044565,0045087,0045944,0050830,0051219,0051607,0060337,0060340,0106310,0140374,0140896,1902554,1904262,1904263,1904417 IC50=8.0nM, Kd=158nM Q9UHD2 23453971 701 GSQSTSNHLWLLSDILGQGATANVFRGRHKKTGDLFAIKVFNNISFLRPVDVQMREFEVLKKLNHKNIVKLFAIEEETTTRHKVLIMEFCPCGSLYTVLEEPSNAYGLPESEFLIVLRDVVGGMNHLRENGIVHRNIKPGNIMRVIGEDGQSVYKLTDFGAARELEDDEQFVSLYGTEEYLHPDMYERAVLRKDHQKKYGATVDLWSIGVTFYHAATGSLPFRPFEGPRRNKEVMYKIITGKPSGAISGVQKAENGPIDWSGDMPVSCSLSRGLQVLLTPVLANILEADQEKCWGFDQFFAETSDILHRMVIHVFSLQQMTAHKIYIHSYNTATIFHELVYKQTKIISSNQELIYEGRRLVLEPGRLAQHFPKTTEENPIFVVSREPLNTIGLIYEKISLPKVHPRYDLDGDASMAKAITGVVCYACRIASTLLLYQELMRKGIRWLIELIKDDYNETVHKKTEVVITLDFCIRNIEKTVKVYEKLGEISDIHTKLLRLSSSQGTIETSLQDIDSRLSPGGSLADAWAHQEGTHPKDRNVEKLQVLLNCMTEIYYQFKKDKAERRLAYNEEQIHKFDKQKLYYHATKAMTHFTDECVKKYEAFLNKSEEWIRKMLHLRKQLLSLTNQCFDIEEEVSKYQEYTNELQET