4ivb A 1.9 BS01 1J5 A 1 L881 V889 A906 M956 F958 L959 S963 E966 L1010 D1021 L29 V37 A54 M95 F97 L98 S102 E105 L149 D160 D1003 A1005 R1007 N1008 D1021 D1040 D142 A144 R146 N147 D160 D179 2.7.10.2 0004672,0004713,0005524,0006468 Ki=1.9nM -logKd/Ki=8.72, Ki=1.9nM EC50=130nM, Ki=1.9nM P23458 23659214 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK