4iti A 2.86 BS01 1HW A 1 A64 M67 V76 L78 L90 M92 H136 I154 A155 D156 L157 S161 F162 A57 M60 V69 L71 L83 M85 H129 I147 A148 D149 L150 S154 F155 D138 K140 E142 N143 D156 T189 D131 K133 E135 N136 D149 T172 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=6.36, IC50=439.5nM Q13546 23473668 301 NVIKMKSSDFLESAELDSGGFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELGGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE