4ibm A 1.8 BS01 IR1 A 1 L1002 G1003 A1028 M1076 E1077 M1079 A1080 G1082 M1139 D1150 L21 G22 A47 M95 E96 M98 A99 G101 M158 D169 D1132 A1134 R1136 N1137 D1150 E1159 L1171 D151 A153 R155 N156 D169 E178 L190 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=1.8uM -logKd/Ki=5.74, IC50=1.8uM P06213 23935097 1301 SVYVPDEWEVSREKITLLRELGQGSFGMVYEGNARDIIKGEAETRVAVKTVNESASLRERIEFLNEASVMKGFTCHHVVRLLGVVSKGQPTLVVMELMAHGDLKSYLRSLRPEAENNPGRPPPTLQEMIQMAAEIADGMAYLNAKKFVHRDLAARNCMVAHDFTVKIGDFGMTRDIYETDYYRKGGKGLLPVRWMAPESLKDGVFTTSSDMWSFGVVLWEITSLAEQPYQGLSNEQVLKFVMDGGYLDQPDNCPERVTDLMRMCWQFNPNMRPTFLEIVNLLKDDLHPSFPEVSFFHSEEN