4gg5 A 2.423 BS01 0J3 A 1 I1084 L1157 Y1159 M1160 R1208 N1209 M1211 A1221 D1222 Y1230 I21 L87 Y89 M90 R138 N139 M141 A151 D152 Y160 D1204 A1206 R1208 N1209 D1222 A1243 D134 A136 R138 N139 D152 A173 2.7.10.1 0004672,0004713,0005524,0006468 ic50=0.93nM -logKd/Ki=9.03, IC50=0.93nM IC50=0.930000nM P08581 22985853 1401 QAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLDNDGKKIHCAVKSLNRITDIQFLTEGIIMKDFSHPNVLSLLGICLRSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKYLASKKFVHRDLAARNCMLDEKFTVKVADFGLARDMYDKEYYSVHNKTGAKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTF