4fz6 A 1.85 BS01 0VG A 1 V385 A400 M450 A451 E452 G454 L501 V21 A36 M81 A82 E83 G85 L132 D494 A496 R498 N499 D512 K533 D125 A127 R129 N130 D143 K160 2.7.10.2 0004672,0004713,0005524,0006468 ic50=127nM -logKd/Ki=6.90, IC50=127nM IC50=127nM P43405 23151054 701 VYLDRKLLTLEDKELGSFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEGHH