4ft5 A 2.4 BS01 H2K A 1 L15 A36 K38 V68 L84 E85 Y86 C87 G90 E91 L137 D148 L13 A29 K31 V53 L69 E70 Y71 C72 G75 E76 L122 D133 D130 K132 E134 N135 D148 T170 D115 K117 E119 N120 D133 T155 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=25nM, IC50=27nM O14757 300 VPFVEDWDLVQTLGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS