4ehz A 2.174 BS01 JAK A 1 V889 A906 M956 F958 L959 E966 L1010 V32 A49 M94 F96 L97 E104 L148 D1003 A1005 R1007 N1008 D1021 D1040 D141 A143 R145 N146 D159 D178 2.7.10.2 0004672,0004713,0005524,0006468 Ki=10nM -logKd/Ki=8.00, Ki=10nM EC50=250nM, Ki=10.0nM P23458 22698084 1201 EKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEDGGNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK