4ehe A 3.3 BS01 RI8 A 1 V471 A481 K483 L505 L514 T529 W531 C532 F583 D594 F595 G596 V24 A34 K36 L58 L67 T82 W84 C85 F136 D147 F148 G149 D576 K578 N580 N581 D594 S616 D129 K131 N133 N134 D147 S159 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.49, IC50=3.2nM P15056 22335519 801 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSLPK