4e4n A 1.9 BS01 0NL A 1 L881 E883 G887 K888 V889 A906 M956 F958 L959 L1010 L29 E31 G35 K36 V37 A54 M95 F97 L98 L149 D1003 A1005 R1007 N1008 D1021 D1040 D142 A144 R146 N147 D160 D179 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.9nM -logKd/Ki=9.05, Ki=0.9nM EC50=91nM, Ki=0.9nM P23458 22591402 1201 GDIVSEKKPATEVDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK