4dgm A 1.65 BS01 AGI A 1 V45 I66 K68 F113 V116 N118 M163 I174 D175 V39 I60 K62 F107 V110 N112 M157 I168 D169 D156 K158 N161 D175 S194 D150 K152 N155 D169 S188 2.7.11.1 0004672,0004674,0005524,0005634,0005829,0005956,0006338,0006468,0016310,0043231,0044024,0051726,0106310 ic50=1.2uM -logKd/Ki=5.92, IC50=1.2uM P28523 22794353 406 SKARVYADVNVLRPKEYWDYEALTVQWGEQDDYEVVRKVGRGKYSEVFEGINVNNNEKCIIKILKPVKKKKIKREIKILQNLMGGPNIVKLLDIVRDQHSKTPSLIFEYVNNTDFKVLYPTLTDYDIRYYIYELLKALDYCHSQGIMHRDVKPHNVMIDHELRKLRLIDWGLAEFYHPGKEYNVRVASRYFKGPELLVDLQDYDYSLDMWSLGCMFAGMIFRKEPFFYGHDNHDQLVKIAKVLGTDGLNVYLNKYRIELDPQLEALVGRHSRKPWLKFMNADNQHLVSPEAIDFLDKLLRYDHQERLTALEAMTHPYFQQVRAAEN