4dbn A 3.15 BS01 0JA A 1 A480 K482 E500 L504 T507 L513 I526 T528 W530 C531 G533 F582 G592 D593 F594 A34 K36 E54 L58 T61 L67 I80 T82 W84 C85 G87 F136 G146 D147 F148 D575 K577 N579 N580 D593 S615 D129 K131 N133 N134 D147 S152 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.15, IC50=7.0nM P15056 22376051 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARSL