4c68 A 1.38 BS01 EN5 A 1 V96 D98 F105 T197 Y211 H213 S215 F226 Y242 G382 G384 D385 G386 V70 D72 F79 T171 Y185 H187 S189 F200 Y216 G356 G358 D359 G360 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0018008,0046872 -logKd/Ki=6.17, IC50=0.68uM A5K1A2 25230674 1000 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4c68 A 1.38 BS02 NHW A 1 Y28 K29 F30 W31 Y95 V96 V160 N161 L163 C164 V165 R170 S171 R173 A175 T183 I186 W192 Q193 A194 Y196 T197 A198 L202 Y393 Y2 K3 F4 W5 Y69 V70 V134 N135 L137 C138 V139 R144 S145 R147 A149 T157 I160 W166 Q167 A168 Y170 T171 A172 L176 Y367 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0018008,0046872 A5K1A2 25230674 1411 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL 4c68 A 1.38 BS03 MG A 1 R170 S171 K172 L174 R144 S145 K146 L148 N161 F162 L163 T197 L410 N135 F136 L137 T171 L384 2.3.1.97 0004379,0005737,0006499,0016746,0018008,0046872 A5K1A2 25230674 1413 DYKFWYTQPVPKINDEFNESVNEPFISDNKVEDVRKDEYKLPPGYSWYVCDVKDEKDRSEIYTLLTDNYVEDDDNIFRFNYSAEFLLWALTSPNYLKTWHIGVKYDASNKLIGFISAIPTDICIHKRTIKMAEVNFLCVHKTLRSKRLAPVLIKEITRRINLENIWQAIYTAGVYLPKPVSDARYYHRSINVKKLIEIGFSSLNSRLTMSRAIKLYRVEDTLNIKNMRLMKKKDVEGVHKLLGSYLEQFNLYAVFTKEEIAHWFLPIENVIYTYVNEENGKIKDMISFYSLPSQILGNDKYSTLNAAYSFYNVTTTATFKQLMQDAILLAKRNNFDVFNALEVMQNKSVFEDLKFGEGDGSLKYYLYNWKCASFAPAHVGIVLL